Kisspeptin-10 vs Selank

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

Kisspeptin-10Selank
CategoryPeptidesPeptides
Standard DoseResearch indicates 1-10 mcg/kg via subcutaneous injection or IV bolus for acute HPG axis stimulation.Research indicates 250-500 mcg daily via intranasal administration (0.15% solution, 2-3 drops per nostril).
TimingMorning dosing preferred for testosterone optimization. Can be used acutely before sexual activity.Can be dosed morning through evening. Unlike Semax, Selank is calming and can be used at night.
Cycle DurationShort-term use only. Continuous kisspeptin administration may cause tachyphylaxis (desensitization) of the HPG axis.14-21 day cycles with equal rest periods.
Evidence Levelmoderate_humanmoderate_human
A

Kisspeptin-10

Peptides

Mechanism

Kisspeptin-10 is the 10-amino acid C-terminal fragment of the kisspeptin family that signals directly to GnRH neurons through the kisspeptin receptor (KISS1R/GPR54), triggering GnRH release into the portal circulation. This stimulates LH and FSH secretion from anterior pituitary gonadotrophs. In men, intravenous kisspeptin-10 produces rapid dose-dependent LH rises (4.1 to 12.4 IU/L at 1 mcg/kg within 30 minutes), increases LH pulse frequency and amplitude, and subsequently elevates testosterone through the HPG axis.

Standard Dosing

Research indicates 1-10 mcg/kg via subcutaneous injection or IV bolus for acute HPG axis stimulation.

Timing

Morning dosing preferred for testosterone optimization. Can be used acutely before sexual activity.

Cycle Duration

Short-term use only. Continuous kisspeptin administration may cause tachyphylaxis (desensitization) of the HPG axis.

Side Effects

  • Facial flushing
  • Mild nausea
  • Elevated LH/testosterone (desired effect)
  • Potential for HPG axis desensitization with prolonged use

Contraindications

  • Hormone-sensitive cancers (prostate, breast)
  • Pregnancy and breastfeeding
  • Children/adolescents (premature puberty risk)

Best Stacking Partners

PT-141HCG
B

Selank

Peptides

Mechanism

Selank (Thr-Lys-Pro-Arg-Pro-Gly-Pro) is a synthetic heptapeptide analog of the immunomodulatory peptide tuftsin (from IgG heavy chain) with a Pro-Gly-Pro extension for metabolic stability. It allosterically modulates GABA-A receptors, enhancing GABA binding and GABAergic neurotransmission. Selank modifies mRNA levels of 84 genes involved in GABAergic neurotransmission in the frontal cortex, enhances enkephalinase inhibition (increasing endogenous enkephalin levels), and modulates serotonergic and noradrenergic systems to produce anxiolytic and nootropic effects.

Standard Dosing

Research indicates 250-500 mcg daily via intranasal administration (0.15% solution, 2-3 drops per nostril).

Timing

Can be dosed morning through evening. Unlike Semax, Selank is calming and can be used at night.

Cycle Duration

14-21 day cycles with equal rest periods.

Side Effects

  • Mild nasal irritation
  • Fatigue/sedation (uncommon)
  • Mild headache

Contraindications

  • Pregnancy and breastfeeding
  • Severe hepatic impairment

Best Stacking Partners

SemaxBPC-157Thymosin Alpha-1

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