Peptides

Selank

Evidence: moderate_human

Mechanism of Action

Selank (Thr-Lys-Pro-Arg-Pro-Gly-Pro) is a synthetic heptapeptide analog of the immunomodulatory peptide tuftsin (from IgG heavy chain) with a Pro-Gly-Pro extension for metabolic stability. It allosterically modulates GABA-A receptors, enhancing GABA binding and GABAergic neurotransmission. Selank modifies mRNA levels of 84 genes involved in GABAergic neurotransmission in the frontal cortex, enhances enkephalinase inhibition (increasing endogenous enkephalin levels), and modulates serotonergic and noradrenergic systems to produce anxiolytic and nootropic effects.

Dosing Protocol

Standard: Research indicates 250-500 mcg daily via intranasal administration (0.15% solution, 2-3 drops per nostril).

Maintenance: Research indicates 250 mcg daily intranasally.

Administration: intranasalsubcutaneous

Timing: Can be dosed morning through evening. Unlike Semax, Selank is calming and can be used at night.

Duration: 14-21 day cycles with equal rest periods.

Notes

Selank is approved in Russia as an anxiolytic and nootropic. Its dual mechanism — GABAergic anxiolysis plus tuftsin-derived immunomodulation — makes it unique among peptide nootropics. It enhances diazepam's anxiolytic effects in research models, suggesting true GABAergic activity. The cognitive stack (Semax + Selank) is widely used in the biohacking community with consistent reports of reduced anxiety plus enhanced focus. Selank is better tolerated than Semax for anxiety-prone individuals.

Stacking

  • Semax
  • BPC-157
  • Thymosin Alpha-1

Interactions

  • Semax [LOW] — Synergistic — the cognitive stack: Semax for focus, Selank for calm. Complementary mechanisms.
  • Benzodiazepines [MEDIUM] — Additive GABAergic effects; Selank enhances diazepam's anxiolytic effects in research.
  • Alcohol [MEDIUM] — Both modulate GABA system; potential for enhanced sedation.

Contraindications

  • Pregnancy and breastfeeding
  • Severe hepatic impairment

Side Effects

  • Mild nasal irritation
  • Fatigue/sedation (uncommon)
  • Mild headache

Key Papers

  • 10.3389/fphar.2016.00031
  • 10.3389/fphar.2017.00089

Source Quality

Russian pharmaceutical-grade (approved in Russia). Research-grade suppliers internationally. Pre-made nasal spray preferred.

Disclaimer: This information is for educational purposes only and is not medical advice. BioAccelera Labs does not diagnose, treat, or prescribe. Consult a licensed healthcare provider before using any compound.

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