Epitalon (Epithalon) vs SS-31 (Elamipretide)

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

✅ Stacking Partners — These compounds are commonly used together and may have synergistic effects.
Epitalon (Epithalon)SS-31 (Elamipretide)
CategoryPeptidesPeptides
Standard DoseResearch indicates 5-10 mg daily via subcutaneous injection for 10-20 day cycles.Research indicates 0.05-0.25 mg/kg daily via subcutaneous injection. Clinical trials used 4-40 mg/day IV or SC.
TimingEvening administration preferred (aligns with pineal/melatonin function). Some protocols split doses AM/PM.Morning dosing preferred. No food timing restrictions.
Cycle Duration10-20 day intensive cycles repeated every 4-6 months. Not used continuously.Clinical trials ranged from single dose to 48 weeks. Optimal cycle length not established.
Evidence Levelanimal_plus_anecdotalEmerging (Phase 2/3 trials)

Mechanism

Epitalon (Ala-Glu-Asp-Gly / AEDG) is a synthetic tetrapeptide based on the natural pineal gland peptide epithalamin. It activates telomerase by inducing expression of the catalytic subunit hTERT, resulting in telomere elongation averaging 33.3% in human somatic cells. Epitalon restores pineal melatonin synthesis and circadian gene expression in aged organisms, increases BDNF, and upregulates CREB1. It also modulates the neuroendocrine system through its effects on the hypothalamic-pituitary axis and antioxidant enzyme regulation.

Standard Dosing

Research indicates 5-10 mg daily via subcutaneous injection for 10-20 day cycles.

Timing

Evening administration preferred (aligns with pineal/melatonin function). Some protocols split doses AM/PM.

Cycle Duration

10-20 day intensive cycles repeated every 4-6 months. Not used continuously.

Side Effects

  • Injection site irritation
  • Mild drowsiness (evening dosing)
  • Vivid dreams

Contraindications

  • Active cancer (telomerase activation concern)
  • History of cancer within 5 years
  • Pregnancy and breastfeeding

Best Stacking Partners

GHK-CuMOTS-cHumanin

Mechanism

SS-31 (D-Arg-Dmt-Lys-Phe-NH2, also known as elamipretide/Bendavia) is a cell-permeable tetrapeptide that localizes to the inner mitochondrial membrane and binds cardiolipin via electrostatic interactions. This stabilizes cardiolipin against oxidative damage, preserving cristae integrity, reducing ROS production, and maintaining mitochondrial ATP production. SS-31 interacts with proteins in two functional groups: oxidative phosphorylation complexes and 2-oxoglutarate metabolic enzymes — all known cardiolipin binders. It restores mitochondrial function without acting as a direct antioxidant.

Standard Dosing

Research indicates 0.05-0.25 mg/kg daily via subcutaneous injection. Clinical trials used 4-40 mg/day IV or SC.

Timing

Morning dosing preferred. No food timing restrictions.

Cycle Duration

Clinical trials ranged from single dose to 48 weeks. Optimal cycle length not established.

Side Effects

  • Injection site reactions
  • Headache
  • Diarrhea (in clinical trials)
  • Nausea

Contraindications

  • Pregnancy and breastfeeding
  • Severe renal impairment (peptide clearance concern)
  • Not commercially available
  • Clinical trial participants only

Best Stacking Partners

MOTS-cHumaninEpitalon

Not sure which is right for you?

Take our free assessment to get personalized recommendations based on your health goals, current stack, and biomarkers.

Get Your Free Protocol →or take the assessment →