Epitalon (Epithalon) vs GHK (without copper)

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

✅ Stacking Partners — These compounds are commonly used together and may have synergistic effects.
Epitalon (Epithalon)GHK (without copper)
CategoryPeptidesPeptides
Standard DoseResearch indicates 5-10 mg daily via subcutaneous injection for 10-20 day cycles.Research indicates 1-3% concentration in topical formulations. Injectable dosing follows GHK-Cu protocols at 1-2 mg daily.
TimingEvening administration preferred (aligns with pineal/melatonin function). Some protocols split doses AM/PM.Topical application morning and evening. Injectable in evening.
Cycle Duration10-20 day intensive cycles repeated every 4-6 months. Not used continuously.Topical use can be ongoing indefinitely. Injectable cycles 8-12 weeks.
Evidence Levelanimal_plus_anecdotalmoderate_human

Mechanism

Epitalon (Ala-Glu-Asp-Gly / AEDG) is a synthetic tetrapeptide based on the natural pineal gland peptide epithalamin. It activates telomerase by inducing expression of the catalytic subunit hTERT, resulting in telomere elongation averaging 33.3% in human somatic cells. Epitalon restores pineal melatonin synthesis and circadian gene expression in aged organisms, increases BDNF, and upregulates CREB1. It also modulates the neuroendocrine system through its effects on the hypothalamic-pituitary axis and antioxidant enzyme regulation.

Standard Dosing

Research indicates 5-10 mg daily via subcutaneous injection for 10-20 day cycles.

Timing

Evening administration preferred (aligns with pineal/melatonin function). Some protocols split doses AM/PM.

Cycle Duration

10-20 day intensive cycles repeated every 4-6 months. Not used continuously.

Side Effects

  • Injection site irritation
  • Mild drowsiness (evening dosing)
  • Vivid dreams

Contraindications

  • Active cancer (telomerase activation concern)
  • History of cancer within 5 years
  • Pregnancy and breastfeeding

Best Stacking Partners

GHK-CuMOTS-cHumanin

Mechanism

GHK (glycyl-L-histidyl-L-lysine) is a naturally occurring tripeptide found in human plasma, saliva, and urine that has an extremely high affinity for copper(II) ions. Even without exogenously complexed copper, GHK rapidly chelates available copper in biological systems, making copper-free GHK functionally similar to GHK-Cu in vivo. The peptide stimulates collagen and glycosaminoglycan synthesis, modulates metalloproteinase activity, resets gene expression patterns toward a healthier state (affecting 31.2% of human genes), and activates wound healing cascades.

Standard Dosing

Research indicates 1-3% concentration in topical formulations. Injectable dosing follows GHK-Cu protocols at 1-2 mg daily.

Timing

Topical application morning and evening. Injectable in evening.

Cycle Duration

Topical use can be ongoing indefinitely. Injectable cycles 8-12 weeks.

Side Effects

  • Mild skin irritation (topical)
  • Injection site reactions

Contraindications

  • Wilson's disease
  • Pregnancy and breastfeeding

Best Stacking Partners

GHK-CuBPC-157Epitalon

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