Growth Factors

GHK-Cu

Evidence: moderate_human

Mechanism of Action

GHK-Cu is a naturally occurring copper-binding tripeptide (glycyl-L-histidyl-L-lysine) that modulates gene expression affecting 31.2% of human genes. It activates Wnt/beta-catenin signaling for hair follicle growth, stimulates TGF-beta pathway for tissue remodeling, and promotes collagen and glycosaminoglycan synthesis while modulating metalloproteinase activity. The copper ion serves as a cofactor for enzymes essential to wound healing including superoxide dismutase and lysyl oxidase.

Dosing Protocol

Standard: Research indicates 1-2 mg daily via subcutaneous injection, or topical application at 1-3% concentration in cream/serum.

Maintenance: Research indicates 1 mg daily or every other day for ongoing skin and tissue maintenance.

Administration: subcutaneoustopicalintradermal

Timing: Evening administration preferred for skin rejuvenation (aligns with nocturnal repair cycles). Topical can be applied morning and evening.

Duration: 8-12 weeks for injectable cycles. Topical use can be ongoing.

Notes

GHK-Cu is the cornerstone of the anti-aging stack (Epitalon + GHK-Cu). It was first identified by Loren Pickart in 1973 from human plasma. Gene profiling via the Broad Institute's Connectivity Map showed GHK can reset gene expression patterns toward a healthier state. Topical GHK-Cu has the most human clinical data of any peptide in this class. At 0.01-100 nM, it increases fibroblast production of elastin and collagen.

Stacking

  • Epitalon
  • BPC-157
  • TB-500
  • Thymosin Alpha-1

Interactions

  • Copper supplements [MEDIUM] — Monitor total copper intake; excess copper can be pro-oxidant and hepatotoxic.
  • Zinc supplements [LOW] — Zinc and copper compete for absorption; space dosing by 2+ hours.
  • Retinoids [LOW] — Synergistic for skin rejuvenation when used topically; may increase sensitivity.
  • Coordinate with copper exposure from other sources

Contraindications

  • Wilson's disease or copper metabolism disorders
  • Liver disease
  • Pregnancy and breastfeeding
  • Use caution with copper-overload states

Side Effects

  • Injection site redness
  • Mild stinging with topical application
  • Transient skin warmth

Key Papers

  • 10.1155/2015/648108
  • 10.1038/288715a0
  • Regenerative peptide literature on GHK-Cu

Source Quality

Pharma-grade for injectable; cosmetic-grade acceptable for topical. Third-party COA essential for copper content verification.

Disclaimer: This information is for educational purposes only and is not medical advice. BioAccelera Labs does not diagnose, treat, or prescribe. Consult a licensed healthcare provider before using any compound.

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