Peptides

Dihexa

Evidence: animal_plus_anecdotal

Mechanism of Action

Dihexa (N-hexanoic-Tyr-Ile-(6)-aminohexanoic amide) is an orally active, blood-brain barrier-permeable oligopeptide derived from angiotensin IV. It binds hepatocyte growth factor (HGF) with high affinity, inhibiting HGF dimerization and synergistically promoting c-Met receptor phosphorylation and signaling. Activation of HGF/c-Met drives procognitive effects through increased dendritic arborization, spinogenesis, and synaptogenesis via the PI3K/AKT signaling pathway. Research indicates it is approximately 10 million times more potent than BDNF for new synapse formation.

Dosing Protocol

Standard: Research indicates 10-20 mg daily via oral or sublingual administration.

Maintenance: Research indicates 10 mg daily or every other day.

Administration: oralsublingualsubcutaneousintranasal

Timing: Morning dosing preferred. Can be taken with or without food (orally active).

Duration: 2-4 week cycles with equal rest periods. Long-term safety data is extremely limited.

Notes

Dihexa is one of the most potent nootropic compounds studied, but carries significant theoretical risk due to HGF/c-Met pathway activation — this same pathway is implicated in multiple cancers. The cancer concern is not trivial and should be discussed thoroughly with any client considering Dihexa. Community reports note dramatic improvements in memory formation and emotional depth. The compound was developed at Washington State University for Alzheimer's research. Oral Dihexa (2 mg/kg) reversed scopolamine-induced cognitive deficits in rats within 7 days. Use with extreme caution and only in clients with no cancer history.

Stacking

  • Semax
  • P21
  • NSI-189

Interactions

  • ACE inhibitors/ARBs [MEDIUM] — Dihexa derives from the angiotensin system; theoretical interaction with RAS-modulating drugs.
  • HGF-modulating cancer therapies [HIGH] — HGF/c-Met pathway is implicated in cancer progression; contraindicated with cancer therapy.
  • Blood thinners [LOW] — HGF promotes angiogenesis; theoretical concern.

Contraindications

  • Active cancer (HGF/c-Met pathway promotes tumor growth)
  • Pregnancy and breastfeeding
  • History of cancer

Side Effects

  • Headache
  • Jaw tension
  • Increased emotional sensitivity (anecdotal)
  • Potential for excessive synaptogenesis (theoretical long-term concern)

Key Papers

  • 10.1124/jpet.114.218735
  • 10.3390/ijms22179510

Source Quality

Research-grade supplier only. Not available through standard compounding pharmacies. Requires careful sourcing with third-party testing.

Disclaimer: This information is for educational purposes only and is not medical advice. BioAccelera Labs does not diagnose, treat, or prescribe. Consult a licensed healthcare provider before using any compound.

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