Humanin vs Tesamorelin

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

HumaninTesamorelin
CategoryPeptidesPeptides
Standard DoseResearch indicates dosing remains experimental. Animal studies use 1-10 mcg/day equivalents. Human protocols are not established.Research indicates 2 mg administered once daily via subcutaneous injection (FDA-approved dose for HIV lipodystrophy).
TimingNo established timing protocol. Morning dosing suggested for neuroprotective applications.Morning administration on empty stomach. Consistent daily timing recommended.
Cycle DurationExperimental — no established cycle lengths.26+ weeks in clinical trials. Long-term use is common; effects are not sustained after discontinuation.
Evidence Levelanimal_plus_anecdotalStrong (FDA-approved indication), Moderate (longevity)
A

Humanin

Peptides

Mechanism

Humanin is a 24-amino acid mitochondrial-derived peptide encoded by the 16S rRNA gene of mitochondrial DNA. It binds IGFBP-3 with high affinity (via Phe-6), interfering with IGFBP-3 binding to importin-beta and suppressing IGFBP-3-mediated apoptosis. It also inhibits the pro-apoptotic protein Bax (Bcl-2 family), preventing mitochondrial outer membrane permeabilization and intrinsic apoptosis. Humanin and IGFBP-3 synergistically protect neurons from amyloid-beta-induced apoptosis, and it activates the STAT3 and ERK1/2 pathways for cytoprotection.

Standard Dosing

Research indicates dosing remains experimental. Animal studies use 1-10 mcg/day equivalents. Human protocols are not established.

Timing

No established timing protocol. Morning dosing suggested for neuroprotective applications.

Cycle Duration

Experimental — no established cycle lengths.

Side Effects

  • Limited data on side effects in humans
  • Theoretical: interference with normal apoptotic processes

Contraindications

  • Active cancer (anti-apoptotic effects could support tumor survival)
  • Pregnancy and breastfeeding

Best Stacking Partners

MOTS-cEpitalonSS-31
B

Tesamorelin

Peptides

Mechanism

Tesamorelin is an FDA-approved synthetic 44-amino acid GHRH analog with a trans-3-hexenoic acid modification at the N-terminal tyrosine that confers resistance to DPP-IV degradation. It binds GHRH receptors on anterior pituitary somatotrophs, stimulating endogenous GH production and secretion while maintaining pulsatile release patterns. Tesamorelin selectively reduces visceral adipose tissue (15-20% reduction in trials) while preserving subcutaneous fat, and markedly increases plasma GH and IGF-1 levels with once-daily dosing.

Standard Dosing

Research indicates 2 mg administered once daily via subcutaneous injection (FDA-approved dose for HIV lipodystrophy).

Timing

Morning administration on empty stomach. Consistent daily timing recommended.

Cycle Duration

26+ weeks in clinical trials. Long-term use is common; effects are not sustained after discontinuation.

Side Effects

  • Injection site reactions (erythema, pruritus)
  • Arthralgia
  • Peripheral edema
  • Myalgia
  • Paresthesia
  • Elevated blood glucose

Contraindications

  • Active cancer or pituitary tumors
  • Pregnancy (Category X)
  • Hypersensitivity to GHRH analogs
  • Disruption of hypothalamic-pituitary axis from surgery/radiation
  • Active cancer
  • Pregnancy
  • Pituitary surgery or disease

Best Stacking Partners

IpamorelinAOD-9604

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