5-Amino-1MQ vs Humanin

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

5-Amino-1MQHumanin
CategoryPeptidesPeptides
Standard DoseResearch indicates 50-150 mg daily via oral administration, typically divided into 1-2 doses.Research indicates dosing remains experimental. Animal studies use 1-10 mcg/day equivalents. Human protocols are not established.
TimingMorning dosing preferred. Can be taken with or without food.No established timing protocol. Morning dosing suggested for neuroprotective applications.
Cycle Duration8-12 week cycles.Experimental — no established cycle lengths.
Evidence Levelanimal_plus_anecdotalanimal_plus_anecdotal
A

5-Amino-1MQ

Peptides

Mechanism

5-Amino-1MQ is a small molecule inhibitor of nicotinamide N-methyltransferase (NNMT), an enzyme that catalyzes the transfer of a methyl group from S-adenosylmethionine (SAM) to nicotinamide, generating 1-methylnicotinamide (1-MNA). By inhibiting NNMT, 5-Amino-1MQ increases intracellular NAD+ levels, reduces 1-MNA production, suppresses lipogenesis in adipocytes, and modulates the methionine-homocysteine cycle. In vivo, it significantly reduces body weight, white adipose mass, and adipocyte size through enhanced energy expenditure and altered lipid metabolism.

Standard Dosing

Research indicates 50-150 mg daily via oral administration, typically divided into 1-2 doses.

Timing

Morning dosing preferred. Can be taken with or without food.

Cycle Duration

8-12 week cycles.

Side Effects

  • Mild GI discomfort
  • Headache
  • Diarrhea (uncommon)
  • Nausea at higher doses

Contraindications

  • Pregnancy and breastfeeding
  • Severe hepatic impairment
  • Active cancer (NAD+ modulation concern)

Best Stacking Partners

MOTS-cAOD-9604TesofensineSemaglutide
B

Humanin

Peptides

Mechanism

Humanin is a 24-amino acid mitochondrial-derived peptide encoded by the 16S rRNA gene of mitochondrial DNA. It binds IGFBP-3 with high affinity (via Phe-6), interfering with IGFBP-3 binding to importin-beta and suppressing IGFBP-3-mediated apoptosis. It also inhibits the pro-apoptotic protein Bax (Bcl-2 family), preventing mitochondrial outer membrane permeabilization and intrinsic apoptosis. Humanin and IGFBP-3 synergistically protect neurons from amyloid-beta-induced apoptosis, and it activates the STAT3 and ERK1/2 pathways for cytoprotection.

Standard Dosing

Research indicates dosing remains experimental. Animal studies use 1-10 mcg/day equivalents. Human protocols are not established.

Timing

No established timing protocol. Morning dosing suggested for neuroprotective applications.

Cycle Duration

Experimental — no established cycle lengths.

Side Effects

  • Limited data on side effects in humans
  • Theoretical: interference with normal apoptotic processes

Contraindications

  • Active cancer (anti-apoptotic effects could support tumor survival)
  • Pregnancy and breastfeeding

Best Stacking Partners

MOTS-cEpitalonSS-31

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