Dihexa vs GHRP-2

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

DihexaGHRP-2
CategoryPeptidesPeptides
Standard DoseResearch indicates 10-20 mg daily via oral or sublingual administration.Research indicates 100-300 mcg administered 1-3 times daily via subcutaneous injection.
TimingMorning dosing preferred. Can be taken with or without food (orally active).On empty stomach, bedtime administration preferred. Wait 2+ hours after last meal.
Cycle Duration2-4 week cycles with equal rest periods. Long-term safety data is extremely limited.8-16 week cycles.
Evidence Levelanimal_plus_anecdotalmoderate_human
A

Dihexa

Peptides

Mechanism

Dihexa (N-hexanoic-Tyr-Ile-(6)-aminohexanoic amide) is an orally active, blood-brain barrier-permeable oligopeptide derived from angiotensin IV. It binds hepatocyte growth factor (HGF) with high affinity, inhibiting HGF dimerization and synergistically promoting c-Met receptor phosphorylation and signaling. Activation of HGF/c-Met drives procognitive effects through increased dendritic arborization, spinogenesis, and synaptogenesis via the PI3K/AKT signaling pathway. Research indicates it is approximately 10 million times more potent than BDNF for new synapse formation.

Standard Dosing

Research indicates 10-20 mg daily via oral or sublingual administration.

Timing

Morning dosing preferred. Can be taken with or without food (orally active).

Cycle Duration

2-4 week cycles with equal rest periods. Long-term safety data is extremely limited.

Side Effects

  • Headache
  • Jaw tension
  • Increased emotional sensitivity (anecdotal)
  • Potential for excessive synaptogenesis (theoretical long-term concern)

Contraindications

  • Active cancer (HGF/c-Met pathway promotes tumor growth)
  • Pregnancy and breastfeeding
  • History of cancer

Best Stacking Partners

SemaxP21NSI-189
B

GHRP-2

Peptides

Mechanism

GHRP-2 (Growth Hormone Releasing Peptide-2) is a synthetic hexapeptide GHS-R1a agonist that is the most potent of the GHRP family for GH release. It stimulates pituitary GH secretion through the ghrelin receptor while also modulating hypothalamic GHRH and somatostatin pathways. GHRP-2 increases GH, cortisol, prolactin, and ACTH release, but with less appetite stimulation than GHRP-6. It also has demonstrated anxiolytic properties and sleep-promoting effects.

Standard Dosing

Research indicates 100-300 mcg administered 1-3 times daily via subcutaneous injection.

Timing

On empty stomach, bedtime administration preferred. Wait 2+ hours after last meal.

Cycle Duration

8-16 week cycles.

Side Effects

  • Water retention
  • Moderate hunger increase (less than GHRP-6)
  • Cortisol elevation
  • Prolactin elevation
  • Tingling
  • Vivid dreams

Contraindications

  • Active cancer
  • Cushing's syndrome
  • Hyperprolactinemia
  • Pregnancy and breastfeeding

Best Stacking Partners

CJC-1295 (no DAC)SermorelinBPC-157

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