5-Amino-1MQ vs Hexarelin

Side-by-side comparison of mechanisms, dosing, interactions, and stacking potential.

5-Amino-1MQHexarelin
CategoryPeptidesPeptides
Standard DoseResearch indicates 50-150 mg daily via oral administration, typically divided into 1-2 doses.Research indicates 100-200 mcg administered 1-2 times daily via subcutaneous injection.
TimingMorning dosing preferred. Can be taken with or without food.On empty stomach, bedtime preferred. Avoid prolonged continuous use due to rapid desensitization.
Cycle Duration8-12 week cycles.4-8 week cycles maximum, then 4+ week break. Hexarelin desensitizes faster than other GHRPs.
Evidence Levelanimal_plus_anecdotalmoderate_human
A

5-Amino-1MQ

Peptides

Mechanism

5-Amino-1MQ is a small molecule inhibitor of nicotinamide N-methyltransferase (NNMT), an enzyme that catalyzes the transfer of a methyl group from S-adenosylmethionine (SAM) to nicotinamide, generating 1-methylnicotinamide (1-MNA). By inhibiting NNMT, 5-Amino-1MQ increases intracellular NAD+ levels, reduces 1-MNA production, suppresses lipogenesis in adipocytes, and modulates the methionine-homocysteine cycle. In vivo, it significantly reduces body weight, white adipose mass, and adipocyte size through enhanced energy expenditure and altered lipid metabolism.

Standard Dosing

Research indicates 50-150 mg daily via oral administration, typically divided into 1-2 doses.

Timing

Morning dosing preferred. Can be taken with or without food.

Cycle Duration

8-12 week cycles.

Side Effects

  • Mild GI discomfort
  • Headache
  • Diarrhea (uncommon)
  • Nausea at higher doses

Contraindications

  • Pregnancy and breastfeeding
  • Severe hepatic impairment
  • Active cancer (NAD+ modulation concern)

Best Stacking Partners

MOTS-cAOD-9604TesofensineSemaglutide
B

Hexarelin

Peptides

Mechanism

Hexarelin (Examorelin) is a synthetic hexapeptide GHS-R1a agonist and the most potent synthetic GH secretagogue by peak GH release. It stimulates GH release through both pituitary ghrelin receptors and hypothalamic pathways, with mechanisms involving regulation of GHRH and somatostatin. Hexarelin also demonstrates significant cardiac benefits through activation of cardiac GHS-R1a receptors, protecting against ischemia-reperfusion injury and reducing cardiac fibrosis via the CD36 scavenger receptor pathway.

Standard Dosing

Research indicates 100-200 mcg administered 1-2 times daily via subcutaneous injection.

Timing

On empty stomach, bedtime preferred. Avoid prolonged continuous use due to rapid desensitization.

Cycle Duration

4-8 week cycles maximum, then 4+ week break. Hexarelin desensitizes faster than other GHRPs.

Side Effects

  • Significant cortisol elevation
  • Prolactin increase
  • Water retention
  • Joint pain
  • Rapid desensitization (unique to Hexarelin)

Contraindications

  • Active cancer
  • Cardiac arrhythmias (due to direct cardiac receptor activity)
  • Cushing's syndrome
  • Pregnancy and breastfeeding

Best Stacking Partners

CJC-1295 (no DAC)Sermorelin

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